PF 477736

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产品编号:P293850

产品规格:100 mg

产品价格:面议


产品详情

标准品编号: P293850
名称: PF 477736
别名: (αR)-α-Amino-N-[5,6-dihydro-2-(1-methyl-1H-pyrazol-4-yl)-6-oxo-1H-pyrrolo[4,3,2-ef][2,3]benzodiazepin-8-yl]cyclohexaneacetamide;
CAS号: 952021-60-2
分子式: C₂₂H₂₅N₇O₂
分子量: 419.48
类别: Research Tools;
应用: P293850 is a selective checkpoint kinase 1 (Chk1) inhibitor (Ki values are 0.49 and 47 nM for Chk1 and Chk2 respectively). Abrogates cell cycle arrest at S and G2-M checkpoints; sensitizes cells to DNA damage.
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