产品编号:P293850
产品规格:100 mg
产品价格:面议
| 标准品编号: | P293850 |
| 名称: | PF 477736 |
| 别名: | (αR)-α-Amino-N-[5,6-dihydro-2-(1-methyl-1H-pyrazol-4-yl)-6-oxo-1H-pyrrolo[4,3,2-ef][2,3]benzodiazepin-8-yl]cyclohexaneacetamide; |
| CAS号: | 952021-60-2 |
| 分子式: | C₂₂H₂₅N₇O₂ |
| 分子量: | 419.48 |
| 类别: | Research Tools; |
| 应用: | P293850 is a selective checkpoint kinase 1 (Chk1) inhibitor (Ki values are 0.49 and 47 nM for Chk1 and Chk2 respectively). Abrogates cell cycle arrest at S and G2-M checkpoints; sensitizes cells to DNA damage. |
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