产品编号：O671020

产品规格：50mg

产品价格：面议

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产品详情

标准品编号:	O671020
名称:	(±)-ORG 28611
别名:	4-[[1-(Cyclohexylmethyl)-7-methoxy-1H-indol-3-yl]carbonyl]-1,2-dimethyl-piperazine; [1-(Cyclohexylmethyl)-7-methoxy-1H-indol-3-yl](3,4-dimethyl-1-piperazinyl)-methanone
CAS号:	784138-08-5
分子式:	C₂₃H₃₃N₃O₂
分子量:	383.53
类别:	Standards; Pharmaceutical/API Drug Impurities/Metabolites;
应用:	(±)-ORG 28611 is full agonist of the human cannabinoid (CB) receptors central CB1 (pEC50 = 7.6; pKi = 8.9) and peripheral CB2 (pKi = 8.8). ORG 28611 (0.1-1 μM/kg, intravenous) demonstrated antinociceptive activity in the mouse tail flick test and the mouse formalin paw test, and it was further evaluated clinically for use as a potential intravenous analgesic agent. Synthetic Cannabinoids
参考文献	Adams, J.M., et al.: Med.Chem.Commun. 1, 54 (2010)