产品编号：C375142
产品规格：2.5mg
产品价格：面议
| 标准品编号: | C375142 |
| 名称: | (S)-2-(4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-N-(4-hydroxyphenyl)acetamide-d4 |
| 别名: | (S)-4-(4-Chlorophenyl)-N-(4-hydroxyphenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetamide-d4; OTX015-d4; |
| 参考CAS: | 202590-98-5 unlabelled |
| 分子式: | C₂₅H₁₈D₄ClN₅O₂S |
| 分子量: | 496.02 |
| 类别: | Standards; Isotopic Labeled Analogues; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites; |
| 应用: | (S)-2-(4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-N-(4-hydroxyphenyl)acetamide-d4 is isotopically labelled (S)-2-(4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-N-(4-hydroxyphenyl)acetamide (C375140), which is an orally bioavailable inhibitor of BRD2, BRD3, BRD4 to AcH4 and shows anti-tumor activity in vitro and in vivo tumor models. |
| 参考文献 | |
