ABT 888

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产品编号:A112580

产品规格:10mg

产品价格:面议


产品详情

标准品编号: A112580
名称: ABT 888
别名: 2-[(2R)-2-Methyl-2-pyrrolidinyl]-1H-benzimidazole-7-carboxamide; A 861695;
CAS号: 912444-00-9
分子式: C₁₃H₁₆N₄O
状态: 白色至Dark Yellow Solid
熔点: >173°C (dec.)
分子量: 244.29
储存: 冰箱保存
溶解性: Methanol (Slightly, Heated), THF (Slightly, Heated)
类别: Research Tools; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites;
应用: ABT-888 is a potent, orally bioavailable PARP-1/-2 inhibitor shown to potentiate DNA damaging agents. The ability to potentiate temozolomide (TMZ) and develop a biological marker for PARP inhibition was evaluated in vivo. Potent PARP inhibitor.
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