Standards; Isotopic Labeled Analogues; Enzyme Activators and Inhibitors;
应用:
THZ1-d6 is isotopically labelled THZ1 (T430000), which is a covalent cyclin-dependent kinases 7 (CDK7) inhibitor. It has the ability to target a remote cysteine residue located outside of the canonical kinase domain, providing a means of achieving selectivity for CDK7.